PDB Information

PDB3CS9
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Characterization of AMN107, a selective inhibitor of native and mutant Bcr-Abl
Weisberg, E., Manley, P.W., Breitenstein, W., Brueggen, J., Cowan-Jacob, S.W., Ray, A., Huntly, B., Fabbro, D., Fendrich, G., Hall-Meyers, E., Kung, A.L., Mestan, J., Daley, G.Q., Callahan, L., Catley, L., Cavazza, C., Azam, M., Neuberg, D., Wright, R.D., Gilliland, D.G., Griffin, J.D.
Cancer Cell
HeaderTransferase
Released2008-04-09
Resolution2.210
CATH Insert Date27 Apr, 2008

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 27 Apr, 2008 Chopped
B 27 Apr, 2008 Chopped
C 27 Apr, 2008 Chopped
D 27 Apr, 2008 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
3cs9A01 01 Apr, 2009 3.30.200.20 Assigned
3cs9A02 01 Apr, 2009 1.10.510.10 Assigned
3cs9B01 01 Apr, 2009 3.30.200.20 Assigned
3cs9B02 01 Apr, 2009 1.10.510.10 Assigned
3cs9C01 01 Apr, 2009 3.30.200.20 Assigned
3cs9C02 01 Apr, 2009 1.10.510.10 Assigned
3cs9D01 01 Apr, 2009 3.30.200.20 Assigned
3cs9D02 01 Apr, 2009 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1