PDB Information

PDB3C1X
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase.
Schroeder, G.M., Chen, X.T., Williams, D.K., Nirschl, D.S., Cai, Z.W., Wei, D., Tokarski, J.S., An, Y., Sack, J., Chen, Z., Huynh, T., Vaccaro, W., Poss, M., Wautlet, B., Gullo-Brown, J., Kellar, K., Manne, V., Hunt, J.T., Wong, T.W., Lombardo, L.J., Fargnoli, J., Borzilleri, R.M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-01-24
Resolution2.170
CATH Insert Date20 Mar, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 20 Mar, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3c1xA01 10 Sep, 2008 3.30.200.20 Assigned
3c1xA02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08581 MET_HUMAN Homo sapiens Hepatocyte growth factor receptor