PDB Information

PDB3APC
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and biological activity of a novel class I PI3K inhibitor, CH5132799
Ohwada, J., Ebiike, H., Kawada, H., Tsukazaki, M., Nakamura, M., Miyazaki, T., Morikami, K., Yoshinari, K., Yoshida, M., Kondoh, O., Kuramoto, S., Ogawa, K., Aoki, Y., Shimma, N.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2010-10-14
Resolution2.540
CATH Insert Date17 Apr, 2011

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 18 Apr, 2011 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
3apcA01 22 Apr, 2011 3.10.20.90 Assigned
3apcA02 22 Apr, 2011 2.60.40.150 Assigned
3apcA03 22 Apr, 2011 1.25.40.70 Assigned
3apcA04 22 Apr, 2011 3.30.1010.10 Assigned
3apcA05 22 Apr, 2011 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform