PDB 2wpa
PDB Information
PDB | 2WPA |
Method | X-RAY DIFFRACTION |
Host Organism | TRICHOPLUSIA NI |
Gene Source | HOMO SAPIENS |
Primary Citation | Optimization of 6,6-Dimethyl Pyrrolo[3,4-C]Pyrazoles: Identification of Pha-793887, a Potent Cdk Inhibitor Suitable for Intravenous Dosing.
Bioorg.Med.Chem.
|
Header | Cell Cycle |
Released | 2009-08-03 |
Resolution | 2.510 |
CATH Insert Date | 25 Feb, 2010 |
PDB Images (13)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 26 Feb, 2010 | Chopped |
B | 26 Feb, 2010 | Chopped |
C | 26 Feb, 2010 | Chopped |
D | 26 Feb, 2010 | Chopped |
CATH Domains (8)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
2wpaA01 | 02 Mar, 2010 | 3.30.200.20 | Assigned |
2wpaA02 | 02 Mar, 2010 | 1.10.510.10 | Assigned |
2wpaB01 | 02 Mar, 2010 | 1.10.472.10 | Assigned |
2wpaB02 | 02 Mar, 2010 | 1.10.472.10 | Assigned |
2wpaC01 | 02 Mar, 2010 | 3.30.200.20 | Assigned |
2wpaC02 | 02 Mar, 2010 | 1.10.510.10 | Assigned |
2wpaD01 | 02 Mar, 2010 | 1.10.472.10 | Assigned |
2wpaD02 | 02 Mar, 2010 | 1.10.472.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P24941 | CDK2_HUMAN | Homo sapiens | Cyclin-dependent kinase 2 |
P24941 | CDK2_HUMAN | Homo sapiens | Cyclin-dependent kinase 2 |
P20248 | CCNA2_HUMAN | Homo sapiens | Cyclin-A2 |
P20248 | CCNA2_HUMAN | Homo sapiens | Cyclin-A2 |