PDB Information

PDB2V4L
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Targeted Polypharmacology: Discovery of Dual Inhibitors of Tyrosine and Phosphoinositide Kinases.
Apsel, B., Blair, J.A., Gonzalez, B., Nazif, T.M., Feldman, M.E., Aizenstein, B., Hoffman, R., Williams, R.L., Shokat, K.M., Knight, Z.A.
Nat.Chem.Biol.
HeaderTransferase
Released2008-09-25
Resolution2.500
CATH Insert Date16 Oct, 2008

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Oct, 2008 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
2v4lA01 17 Oct, 2008 3.10.20.90 Assigned
2v4lA02 17 Oct, 2008 2.60.40.150 Assigned
2v4lA03 17 Oct, 2008 1.25.40.70 Assigned
2v4lA04 17 Oct, 2008 3.30.1010.10 Assigned
2v4lA05 17 Oct, 2008 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform