PDB Information

PDB2R9S
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
3,5-Disubstituted quinolines as novel c-Jun N-terminal kinase inhibitors.
Jiang, R., Duckett, D., Chen, W., Habel, J., Ling, Y.Y., LoGrasso, P., Kamenecka, T.M.
Bioorg.Med.Chem.Lett.
HeaderSignaling Protein, Transferase
Released2007-09-13
Resolution2.400
CATH Insert Date07 Nov, 2007

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Nov, 2007 Chopped
B 08 Nov, 2007 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2r9sA01 23 Nov, 2007 3.30.200.20 Assigned
2r9sA02 23 Nov, 2007 1.10.510.10 Assigned
2r9sB01 23 Nov, 2007 3.30.200.20 Assigned
2r9sB02 23 Nov, 2007 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P53779 MK10_HUMAN Homo sapiens Mitogen-activated protein kinase 10
P53779 MK10_HUMAN Homo sapiens Mitogen-activated protein kinase 10