PDB Information

PDB2R2L
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Efficacy, pharmacokinetics, and metabolism of tetrahydroquinoline inhibitors of Plasmodium falciparum protein farnesyltransferase.
Van Voorhis, W.C., Rivas, K.L., Bendale, P., Nallan, L., Horney, C., Barrett, L.K., Bauer, K.D., Smart, B.P., Ankala, S., Hucke, O., Verlinde, C.L., Chakrabarti, D., Strickland, C., Yokoyama, K., Buckner, F.S., Hamilton, A.D., Williams, D.K., Lombardo, L.J., Floyd, D., Gelb, M.H.
Antimicrob.Agents Chemother.
HeaderTransferase
Released2007-08-27
Resolution2.230
CATH Insert Date13 Mar, 2008

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 13 Mar, 2008 Chopped
B 13 Mar, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2r2lA00 14 Mar, 2008 1.25.40.120 Assigned
2r2lB00 14 Mar, 2008 1.50.10.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q02293 FNTB_RAT Rattus norvegicus Protein farnesyltransferase subunit beta
Q04631 FNTA_RAT Rattus norvegicus Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha