PDB Information

PDB2QU2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Thiophene substituted acylguanidines as BACE1 inhibitors.
Fobare, W.F., Solvibile, W.R., Robichaud, A.J., Malamas, M.S., Manas, E., Turner, J., Hu, Y., Wagner, E., Chopra, R., Cowling, R., Jin, G., Bard, J.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2007-08-03
Resolution2.600
CATH Insert Date07 Aug, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Aug, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2qu2A01 08 Aug, 2008 2.40.70.10 Assigned
2qu2A02 08 Aug, 2008 2.40.70.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P56817 BACE1_HUMAN Homo sapiens Beta-secretase 1