PDB Information

PDB2QBR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based optimization of protein tyrosine phosphatase 1B inhibitors: from the active site to the second phosphotyrosine binding site.
Wilson, D.P., Wan, Z.K., Xu, W.X., Kirincich, S.J., Follows, B.C., Joseph-McCarthy, D., Foreman, K., Moretto, A., Wu, J., Zhu, M., Binnun, E., Zhang, Y.L., Tam, M., Erbe, D.V., Tobin, J., Xu, X., Leung, L., Shilling, A., Tam, S.Y., Mansour, T.S., Lee, J.
J.Med.Chem.
HeaderHydrolase
Released2007-06-18
Resolution2.300
CATH Insert Date20 Mar, 2008

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 20 Mar, 2008 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
2qbrA00 21 Mar, 2008 3.90.190.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P18031 PTN1_HUMAN Homo sapiens Tyrosine-protein phosphatase non-receptor type 1