PDB Information

PDB2Q8I
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Distinct Structural Mechanisms for Inhibition of Pyruvate Dehydrogenase Kinase Isoforms by AZD7545, Dichloroacetate, and Radicicol.
Kato, M., Li, J., Chuang, J.L., Chuang, D.T.
Structure
HeaderTransferase
Released2007-06-10
Resolution2.600
CATH Insert Date26 Jul, 2007

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 26 Jul, 2007 Chopped
B 26 Jul, 2007 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
2q8iA01 17 Aug, 2007 1.20.140.20 Assigned
2q8iA02 17 Aug, 2007 3.30.565.10 Assigned
2q8iB00 16 Aug, 2007 2.40.50.100 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P10515 ODP2_HUMAN Homo sapiens Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, mitochondrial
Q15120 PDK3_HUMAN Homo sapiens [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial