PDB Information

PDB2Q8H
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Distinct Structural Mechanisms for Inhibition of Pyruvate Dehydrogenase Kinase Isoforms by AZD7545, Dichloroacetate, and Radicicol.
Kato, M., Li, J., Chuang, J.L., Chuang, D.T.
Structure
HeaderTransferase
Released2007-06-10
Resolution2.000
CATH Insert Date26 Jul, 2007

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 26 Jul, 2007 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2q8hA01 17 Aug, 2007 1.20.140.20 Assigned
2q8hA02 17 Aug, 2007 3.30.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q15118 PDK1_HUMAN Homo sapiens [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial