PDB 2pzy
PDB Information
| PDB | 2PZY |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | The discovery of carboline analogs as potent MAPKAP-K2 inhibitors
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2007-05-18 |
| Resolution | 2.900 |
| CATH Insert Date | 07 Nov, 2007 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Nov, 2007 | Chopped |
| B | 08 Nov, 2007 | Chopped |
| C | 08 Nov, 2007 | Chopped |
| D | 08 Nov, 2007 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 2pzyA01 | 10 Sep, 2008 | 3.30.200.20 | Assigned |
| 2pzyA02 | 10 Sep, 2008 | 1.10.510.10 | Assigned |
| 2pzyB01 | 08 Dec, 2008 | 3.30.200.20 | Assigned |
| 2pzyB02 | 08 Dec, 2008 | 1.10.510.10 | Assigned |
| 2pzyC01 | 08 Dec, 2008 | 3.30.200.20 | Assigned |
| 2pzyC02 | 08 Dec, 2008 | 1.10.510.10 | Assigned |
| 2pzyD01 | 08 Dec, 2008 | 3.30.200.20 | Assigned |
| 2pzyD02 | 08 Dec, 2008 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P49137 | MAPK2_HUMAN | Homo sapiens | MAP kinase-activated protein kinase 2 |
| P49137 | MAPK2_HUMAN | Homo sapiens | MAP kinase-activated protein kinase 2 |
| P49137 | MAPK2_HUMAN | Homo sapiens | MAP kinase-activated protein kinase 2 |
| P49137 | MAPK2_HUMAN | Homo sapiens | MAP kinase-activated protein kinase 2 |
