PDB 2p4i
PDB Information
| PDB | 2P4I |
| Method | X-RAY DIFFRACTION |
| Host Organism | Trichoplusia ni |
| Gene Source | Homo sapiens |
| Primary Citation | Evolution of a highly selective and potent 2-(pyridin-2-yl)-1,3,5-triazine Tie-2 kinase inhibitor.
J.Med.Chem.
|
| Header | Transferase |
| Released | 2007-03-12 |
| Resolution | 2.500 |
| CATH Insert Date | 22 Mar, 2007 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 22 Mar, 2007 | Chopped |
| B | 22 Mar, 2007 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 2p4iA01 | 10 Sep, 2008 | 3.30.200.20 | Assigned |
| 2p4iA02 | 10 Sep, 2008 | 1.10.510.10 | Assigned |
| 2p4iB01 | 10 Sep, 2008 | 3.30.200.20 | Assigned |
| 2p4iB02 | 10 Sep, 2008 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q02763 | TIE2_HUMAN | Homo sapiens | Angiopoietin-1 receptor |
| Q02763 | TIE2_HUMAN | Homo sapiens | Angiopoietin-1 receptor |
