PDB Information

PDB2NO3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a new class of 4-anilinopyrimidines as potent c-Jun N-terminal kinase inhibitors: Synthesis and SAR studies.
Liu, M., Wang, S., Clampit, J.E., Gum, R.J., Haasch, D.L., Rondinone, C.M., Trevillyan, J.M., Abad-Zapatero, C., Fry, E.H., Sham, H.L., Liu, G.
Bioorg.Med.Chem.Lett.
HeaderSignaling Protein/Inhibitor
Released2006-10-24
Resolution3.200
CATH Insert Date19 Apr, 2007

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 19 Apr, 2007 Chopped
B 19 Apr, 2007 Chopped
F 19 Apr, 2007 Rejected
G 19 Apr, 2007 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2no3A01 19 Jul, 2007 3.30.200.20 Assigned
2no3A02 19 Jul, 2007 1.10.510.10 Assigned
2no3B01 19 Jul, 2007 3.30.200.20 Assigned
2no3B02 19 Jul, 2007 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8