PDB Information

PDB2G1R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Ketopiperazine-Based Renin Inhibitors: Optimization of the "C" Ring
Holsworth, D.D., Cai, C., Cheng, X.M., Cody, W.L., Downing, D.M., Erasga, N., Lee, C., Powell, N.A., Ednunds, J.J., Stier, M., Jalaie, M., Zhang, E., McConnell, P., Ryan, M.J., Bryant, J., Li, T., Kasani, A., Hall, E., Subedi, R., Rahim, M., Maiti, S.
BIOORG.MED.CHEM.LETT.
HeaderHydrolase
Released2006-02-14
Resolution2.420
CATH Insert Date14 Jul, 2006

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Jul, 2006 Chopped
B 14 Jul, 2006 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2g1rA01 16 Oct, 2006 2.40.70.10 Assigned
2g1rA02 16 Oct, 2006 2.40.70.10 Assigned
2g1rB01 16 Oct, 2006 2.40.70.10 Assigned
2g1rB02 16 Oct, 2006 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00797 RENI_HUMAN Homo sapiens Renin
P00797 RENI_HUMAN Homo sapiens Renin