PDB 2g01
PDB Information
| PDB | 2G01 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Synthesis and SAR of 1,9-dihydro-9-hydroxypyrazolo[3,4-b]quinolin-4-ones as novel, selective c-Jun N-terminal kinase inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2006-02-10 |
| Resolution | 3.500 |
| CATH Insert Date | 14 Jul, 2006 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Jul, 2006 | Chopped |
| B | 14 Jul, 2006 | Chopped |
| F | 14 Jul, 2006 | Rejected |
| G | 14 Jul, 2006 | Rejected |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 2g01A01 | 16 Oct, 2006 | 3.30.200.20 | Assigned |
| 2g01A02 | 16 Oct, 2006 | 1.10.510.10 | Assigned |
| 2g01B01 | 16 Oct, 2006 | 3.30.200.20 | Assigned |
| 2g01B02 | 16 Oct, 2006 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9UQF2 | JIP1_HUMAN | Homo sapiens | C-Jun-amino-terminal kinase-interacting protein 1 |
| P45983 | MK08_HUMAN | Homo sapiens | Mitogen-activated protein kinase 8 |
| Q9UQF2 | JIP1_HUMAN | Homo sapiens | C-Jun-amino-terminal kinase-interacting protein 1 |
| P45983 | MK08_HUMAN | Homo sapiens | Mitogen-activated protein kinase 8 |
