PDB Information

PDB2FLR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Novel 5-azaindole factor VIIa inhibitors.
Riggs, J.R., Hu, H., Kolesnikov, A., Leahy, E.M., Wesson, K.E., Shrader, W.D., Vijaykumar, D., Wahl, T.A., Tong, Z., Sprengeler, P.A., Green, M.J., Yu, C., Katz, B.A., Sanford, E., Nguyen, M., Cabuslay, R., Young, W.B.
Bioorg.Med.Chem.Lett.
HeaderHydrolase/Blood Clotting
Released2006-01-06
Resolution2.350
CATH Insert Date23 Feb, 2007

PDB Images (9)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
H 23 Feb, 2007 Chopped
L 23 Feb, 2007 Chopped
T 23 Feb, 2007 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
2flrH01 24 Jul, 2007 2.40.10.10 Assigned
2flrH02 24 Jul, 2007 2.40.10.10 Assigned
2flrL01 13 Jul, 2007 2.10.25.10 Assigned
2flrL02 13 Jul, 2007 2.10.25.10 Assigned
2flrT00 14 Jul, 2007 2.60.40.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P08709 FA7_HUMAN Homo sapiens Coagulation factor VII
P08709 FA7_HUMAN Homo sapiens Coagulation factor VII
P13726 TF_HUMAN Homo sapiens Tissue factor