PDB Information

PDB2CHM
MethodX-RAY DIFFRACTION
Host OrganismTRICHOPLUSIA NI
Gene SourceHOMO SAPIENS
Primary Citation
A Novel Series of Potent and Selective Pde5 Inhibitors with Potential for High and Dose-Independent Oral Bioavailability
Allerton, C.M.N., Barber, C.G., Beaumont, K.C., Brown, D.G., Cole, S.M., Ellis, D., Lane, C.A.L., Maw, G.N., Mount, N.M., Rawson, D.J., Robinson, C.M., Street, S.D.A., Summerhill, N.W.
J.Med.Chem.
HeaderHydrolase
Released2006-03-15
Resolution1.600
CATH Insert Date14 Jul, 2006

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Jul, 2006 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
2chmA00 15 Oct, 2006 1.10.1300.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q07343 PDE4B_HUMAN Homo sapiens cAMP-specific 3',5'-cyclic phosphodiesterase 4B
O76074 PDE5A_HUMAN Homo sapiens cGMP-specific 3',5'-cyclic phosphodiesterase