PDB Information

PDB2C4G
MethodX-RAY DIFFRACTION
Host OrganismTRICHOPLUSIA NI
Gene SourceHOMO SAPIENS
Primary Citation
3-Amino-1,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazoles: A New Class of Cdk2 Inhibitors.
Pevarello, P., Fancelli, D., Vulpetti, A., Amici, R., Villa, M., Pittala, V., Vianello, P., Cameron, A., Ciomei, M., Mercurio, C., Bischoff, J.R., Roletto, F., Varasi, M., Brasca, M.G.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2005-10-17
Resolution2.700
CATH Insert Date05 Mar, 2006

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped
C 05 Mar, 2006 Chopped
D 05 Mar, 2006 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
2c4gA01 10 Mar, 2006 3.30.200.20 Assigned
2c4gA02 10 Mar, 2006 1.10.510.10 Assigned
2c4gB01 10 Mar, 2006 1.10.472.10 Assigned
2c4gB02 10 Mar, 2006 1.10.472.10 Assigned
2c4gC01 10 Mar, 2006 3.30.200.20 Assigned
2c4gC02 10 Mar, 2006 1.10.510.10 Assigned
2c4gD01 10 Mar, 2006 1.10.472.10 Assigned
2c4gD02 10 Mar, 2006 1.10.472.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2