PDB Information

PDB2BQ6
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Probing the Subpockets of Factor Xa Reveals Two Binding Modes for Inhibitors Based on a 2-Carboxyindole Scaffold: A Study Combining Structure-Activity Relationship and X-Ray Crystallography.
Nazare, M., Will, D.W., Matter, H., Schreuder, H., Ritter, K., Urmann, M., Essrich, M., Bauer, A., Wagner, M., Czech, J., Lorenz, M., Laux, V., Wehner, V.
J.Med.Chem.
HeaderHydrolase
Released2005-04-27
Resolution3.000
CATH Insert Date14 Jul, 2006

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Jul, 2006 Chopped
B 14 Jul, 2006 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
2bq6A00 16 Oct, 2006 2.10.25.10 Assigned
2bq6B01 17 Oct, 2006 2.40.10.10 Assigned
2bq6B02 17 Oct, 2006 2.40.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X