PDB Information

PDB1URC
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Design, synthesis, biological activity and structural analysis of cyclic peptide inhibitors targeting the substrate recruitment site of cyclin-dependent kinase complexes.
Andrews, M.J., McInnes, C., Kontopidis, G., Innes, L., Cowan, A., Plater, A., Fischer, P.M.
Org. Biomol. Chem.
HeaderTransferase/Inhibitor
Released2003-10-28
Resolution2.600
CATH Insert Date05 Mar, 2006

PDB Images (15)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped
C 05 Mar, 2006 Chopped
D 05 Mar, 2006 Chopped
E 05 Mar, 2006 Rejected
F 05 Mar, 2006 Rejected

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
1urcA01 05 Mar, 2006 3.30.200.20 Assigned
1urcA02 05 Mar, 2006 1.10.510.10 Assigned
1urcB01 05 Mar, 2006 1.10.472.10 Assigned
1urcB02 05 Mar, 2006 1.10.472.10 Assigned
1urcC01 18 Jan, 2007 3.30.200.20 Assigned
1urcC02 18 Jan, 2007 1.10.510.10 Assigned
1urcD01 05 Mar, 2006 1.10.472.10 Assigned
1urcD02 05 Mar, 2006 1.10.472.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2