PDB Information

PDB1SZM
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceBos taurus
Primary Citation
The protein kinase C inhibitor bisindolyl maleimide 2 binds with reversed orientations to different conformations of protein kinase a.
Gassel, M., Breitenlechner, C.B., Koenig, N., Huber, R., Engh, R.A., Bossemeyer, D.
J.Biol.Chem.
HeaderTransferase
Released2004-04-06
Resolution2.500
CATH Insert Date05 Mar, 2006

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
1szmA01 05 Mar, 2006 1.10.510.10 Assigned
1szmA02 05 Mar, 2006 3.30.200.20 Assigned
1szmB01 05 Mar, 2006 1.10.510.10 Assigned
1szmB02 05 Mar, 2006 3.30.200.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha