PDB Information

PDB1QXK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Identification of a Monoacid-Based, Cell Permeable, Selective Inhibitor of Protein Tyrosine Phosphatase 1B
Xin, Z., Liu, G., Abad-Zapatero, C., Pei, Z., Szczepankiewick, B.G., Li, X., Zhang, T., Hutchins, C.W., Hajduk, P.J., Ballaron, S.J., Stashko, M.A., Lubben, T.H., Trevillyan, J.M., Jirousek, M.R.
BIOORG.MED.CHEM.LETT.
HeaderHydrolase
Released2003-09-08
Resolution2.300
CATH Insert Date05 Mar, 2006

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
1qxkA00 05 Mar, 2006 3.90.190.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P18031 PTN1_HUMAN Homo sapiens Tyrosine-protein phosphatase non-receptor type 1