PDB Information

PDB1PYN
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery and SAR of novel, potent and selective protein tyrosine phosphatase 1B inhibitors.
Pei, Z., Li, X., Liu, G., Abad-Zapatero, C., Lubben, T., Zhang, T., Ballaron, S.J., Hutchins, C.W., Trevillyan, J.M., Jirousek, M.R.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2003-07-09
Resolution2.200
CATH Insert Date05 Mar, 2006

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
1pynA00 05 Mar, 2006 3.90.190.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P18031 PTN1_HUMAN Homo sapiens Tyrosine-protein phosphatase non-receptor type 1