PDB Information

PDB1KYN
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Nonpeptide inhibitors of cathepsin G: optimization of a novel beta-ketophosphonic acid lead by structure-based drug design.
Greco, M.N., Hawkins, M.J., Powell, E.T., Almond Jr., H.R., Corcoran, T.W., de Garavilla, L., Kauffman, J.A., Recacha, R., Chattopadhyay, D., Andrade-Gordon, P., Maryanoff, B.E.
J.Am.Chem.Soc.
HeaderHydrolase
Released2002-02-05
Resolution3.500
CATH Insert Date05 Mar, 2006

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
1kynA01 05 Mar, 2006 2.40.10.10 Assigned
1kynA02 05 Mar, 2006 2.40.10.10 Assigned
1kynB01 05 Mar, 2006 2.40.10.10 Assigned
1kynB02 05 Mar, 2006 2.40.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P08311 CATG_HUMAN Homo sapiens Cathepsin G
P08311 CATG_HUMAN Homo sapiens Cathepsin G