PDB Information

PDB1GJA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets.
Katz, B.A., Sprengeler, P.A., Luong, C., Verner, E., Elrod, K., Kirtley, M., Janc, J., Spencer, J.R., Breitenbucher, J.G., Hui, H., McGee, D., Allen, D., Martelli, A., Mackman, R.L.
Chem.Biol.
HeaderBlood Clotting, Hydrolase
Released2001-04-27
Resolution1.560
CATH Insert Date05 Mar, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Rejected
B 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1gjaB01 05 Mar, 2006 2.40.10.10 Assigned
1gjaB02 05 Mar, 2006 2.40.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator