CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Retinoic acid receptor RXR-alpha

Enzyme Information

UniProtKB Entries (1)

P19793
RXRA_HUMAN
Homo sapiens
Retinoic acid receptor RXR-alpha

PDB Structure

PDB 4M8E
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Methyl-substituted conformationally constrained rexinoid agonists for the retinoid X receptors demonstrate improved efficacy for cancer therapy and prevention.
Desphande, A., Xia, G., Boerma, L.J., Vines, K.K., Atigadda, V.R., Lobo-Ruppert, S., Grubbs, C.J., Moeinpour, F.L., Smith, C.D., Christov, K., Brouillette, W.J., Muccio, D.D.
Bioorg.Med.Chem.