CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Androgen receptor variant

Enzyme Information

UniProtKB Entries (1)

P10275
ANDR_HUMAN
Homo sapiens
Androgen receptor

PDB Structure

PDB 4HLW
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Targeting the Binding Function 3 (BF3) Site of the Androgen Receptor Through Virtual Screening. 2. Development of 2-((2-phenoxyethyl) thio)-1H-benzimidazole Derivatives.
Munuganti, R.S., Leblanc, E., Axerio-Cilies, P., Labriere, C., Frewin, K., Singh, K., Hassona, M.D., Lack, N.A., Li, H., Ban, F., Tomlinson Guns, E., Young, R., Rennie, P.S., Cherkasov, A.
J.Med.Chem.