PDB Information

PDB6UDY
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an alpha-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere.
Rescourio, G., Gonzalez, A.Z., Jabri, S., Belmontes, B., Moody, G., Whittington, D., Huang, X., Caenepeel, S., Cardozo, M., Cheng, A.C., Chow, D., Dou, H., Jones, A., Kelly, R.C., Li, Y., Lizarzaburu, M., Lo, M.C., Mallari, R., Meleza, C., Rew, Y., Simonovich, S., Sun, D., Turcotte, S., Yan, X., Wong, S.G., Yanez, E., Zancanella, M., Houze, J., Medina, J.C., Hughes, P.E., Brown, S.P.
J.Med.Chem.
HeaderApoptosis/Inhibitor
Released2019-09-19
Resolution1.700
CATH Insert Date15 Dec, 2019

PDB Images (1)

PDB Prints

PDB Chains (0)

Chain ID Date inserted into CATH CATH Status

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description