PDB Information

PDB6UCS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli K-12
Gene SourceHomo sapiens
Primary Citation
Discovery and Structure-Based Optimization of Potent and Selective WD repeat domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core.
Tian, J., Teuscher, K., Aho, E.R., Alvarado, J.R., Mills, J.J., Meyers, K.M., Gogliotti, R.D., Han, C., Macdonald, J.D., Sai, J., Shaw, J.G., Sensintaffar, J.L., Zhao, B., Rietz, T.A., Thomas, L.R., Payne, W.G., Moore, W.J., Stott, G.M., Kondo, J., Inoue, M., Coffey, R., Tansey, W.P., Stauffer, S., Lee, T., Fesik, S.W.
J.Med.Chem.
HeaderTranscription
Released2019-09-17
Resolution1.850
CATH Insert Date05 Jan, 2020

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Chain ID Date inserted into CATH CATH Status

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Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description