PDB Information

PDB6P9F
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Identification of potent, selective and orally bioavailable phenyl ((R)-3-phenylpyrrolidin-3-yl)sulfone analogues as ROR gamma t inverse agonists.
Lu, Z., Duan, J.J., Xiao, H., Neels, J., Wu, D.R., Weigelt, C.A., Sack, J.S., Khan, J., Ruzanov, M., An, Y., Yarde, M., Karmakar, A., Vishwakrishnan, S., Baratam, V., Shankarappa, H., Vanteru, S., Babu, V., Basha, M., Kumar Gupta, A., Kumaravel, S., Mathur, A., Zhao, Q., Salter-Cid, L.M., Carter, P.H., Murali Dhar, T.G.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2019-06-10
Resolution2.800
CATH Insert Date04 Aug, 2019

PDB Images (3)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 04 Aug, 2019 New
B 04 Aug, 2019 New

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description