PDB Information

PDB6OCU
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and optimization of heteroaryl piperazines as potent and selective PI3K delta inhibitors.
Zhou, H., McGowan, M.A., Lipford, K., Christopher, M., Fradera, X., Witter, D., Lesburg, C.A., Li, C., Methot, J.L., Lampe, J., Achab, A., Shaffer, L., Goldenblatt, P., Shah, S., Bass, A., Schroeder, G., Chen, D., Zeng, H., Augustin, M.A., Katz, J.D.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2019-03-25
Resolution2.770
CATH Insert Date15 Dec, 2019

PDB Images (1)

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PDB Chains (0)

Chain ID Date inserted into CATH CATH Status

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description