PDB Information

PDB6MUL
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Structure Overhaul Affords a Potent Purine PI3K delta Inhibitor with Improved Tolerability.
Methot, J.L., Zhou, H., Kattar, S.D., McGowan, M.A., Wilson, K., Garcia, Y., Deng, Y., Altman, M., Fradera, X., Lesburg, C., Fischmann, T., Li, C., Alves, S., Shah, S., Fernandez, R., Goldenblatt, P., Hill, A., Shaffer, L., Chen, D., Tong, V., McLeod, R.L., Yu, H., Bass, A., Kemper, R., Gatto, N.T., LaFranco-Scheuch, L., Trotter, B.W., Guzi, T., Katz, J.D.
J.Med.Chem.
HeaderTransferase
Released2018-10-23
Resolution3.090
CATH Insert Date05 May, 2019

PDB Images (3)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 May, 2019 Holding pen
B 05 May, 2019 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform