PDB Information

PDB6HTY
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and Characterization of the Potent and Selective P2X4 InhibitorN-[4-(3-Chlorophenoxy)-3-sulfamoylphenyl]-2-phenylacetamide (BAY-1797) and Structure-Guided Amelioration of Its CYP3A4 Induction Profile.
Werner, S., Mesch, S., Hillig, R.C., Ter Laak, A., Klint, J., Neagoe, I., Laux-Biehlmann, A., Dahllof, H., Brauer, N., Puetter, V., Nubbemeyer, R., Schulz, S., Bairlein, M., Zollner, T.M., Steinmeyer, A.
J.Med.Chem.
HeaderTranscription
Released2018-10-05
Resolution2.220
CATH Insert Date08 Dec, 2019

PDB Images (1)

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PDB Chains (0)

Chain ID Date inserted into CATH CATH Status

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description