PDB Information

PDB6HTC
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae S288c
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of Inhibitors Selective for Human Proteasome beta 2c or beta 2i Subunits.
Xin, B.T., Huber, E.M., de Bruin, G., Heinemeyer, W., Maurits, E., Espinal, C., Du, Y., Janssens, M., Weyburne, E.S., Kisselev, A.F., Florea, B.I., Driessen, C., van der Marel, G.A., Groll, M., Overkleeft, H.S.
J.Med.Chem.
HeaderHydrolase
Released2018-10-03
Resolution2.800
CATH Insert Date03 Feb, 2019

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 03 Feb, 2019 Chopped
A 03 Feb, 2019 Chopped
b 03 Feb, 2019 Chopped
B 03 Feb, 2019 Chopped
C 03 Feb, 2019 Chopped
D 03 Feb, 2019 Chopped
E 03 Feb, 2019 Chopped
F 03 Feb, 2019 Chopped
G 03 Feb, 2019 Chopped
H 03 Feb, 2019 Chopped
I 03 Feb, 2019 Chopped
J 03 Feb, 2019 Chopped
K 03 Feb, 2019 Chopped
L 03 Feb, 2019 Chopped
M 03 Feb, 2019 Chopped
N 03 Feb, 2019 Chopped
O 03 Feb, 2019 Chopped
P 03 Feb, 2019 Chopped
Q 03 Feb, 2019 Chopped
R 03 Feb, 2019 Chopped
S 03 Feb, 2019 Chopped
T 03 Feb, 2019 Chopped
U 03 Feb, 2019 Chopped
V 03 Feb, 2019 Chopped
W 03 Feb, 2019 Chopped
X 03 Feb, 2019 Chopped
Y 03 Feb, 2019 Chopped
Z 03 Feb, 2019 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
6htca00 04 Feb, 2019 3.60.20.10 Assigned
6htcA00 04 Feb, 2019 3.60.20.10 Assigned
6htcb00 04 Feb, 2019 3.60.20.10 Assigned
6htcB00 04 Feb, 2019 3.60.20.10 Assigned
6htcC00 04 Feb, 2019 3.60.20.10 Assigned
6htcD00 04 Feb, 2019 3.60.20.10 Assigned
6htcE00 04 Feb, 2019 3.60.20.10 Assigned
6htcF00 04 Feb, 2019 3.60.20.10 Assigned
6htcG00 04 Feb, 2019 3.60.20.10 Assigned
6htcH00 04 Feb, 2019 3.60.20.10 Assigned
6htcI00 04 Feb, 2019 3.60.20.10 Assigned
6htcJ00 04 Feb, 2019 3.60.20.10 Assigned
6htcK00 04 Feb, 2019 3.60.20.10 Assigned
6htcL00 04 Feb, 2019 3.60.20.10 Assigned
6htcM00 04 Feb, 2019 3.60.20.10 Assigned
6htcN00 04 Feb, 2019 3.60.20.10 Assigned
6htcO00 04 Feb, 2019 3.60.20.10 Assigned
6htcP00 04 Feb, 2019 3.60.20.10 Assigned
6htcQ00 04 Feb, 2019 3.60.20.10 Assigned
6htcR00 04 Feb, 2019 3.60.20.10 Assigned
6htcS00 04 Feb, 2019 3.60.20.10 Assigned
6htcT00 04 Feb, 2019 3.60.20.10 Assigned
6htcU00 04 Feb, 2019 3.60.20.10 Assigned
6htcV00 04 Feb, 2019 3.60.20.10 Assigned
6htcW00 04 Feb, 2019 3.60.20.10 Assigned
6htcX00 04 Feb, 2019 3.60.20.10 Assigned
6htcY00 04 Feb, 2019 3.60.20.10 Assigned
6htcZ00 04 Feb, 2019 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
Q99436 PSB7_HUMAN Homo sapiens Proteasome subunit beta type-7
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
Q99436 PSB7_HUMAN Homo sapiens Proteasome subunit beta type-7
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5