PDB Information

PDB6GZH
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Small Molecules Co-targeting CKI alpha and the Transcriptional Kinases CDK7/9 Control AML in Preclinical Models.
Minzel, W., Venkatachalam, A., Fink, A., Hung, E., Brachya, G., Burstain, I., Shaham, M., Rivlin, A., Omer, I., Zinger, A., Elias, S., Winter, E., Erdman, P.E., Sullivan, R.W., Fung, L., Mercurio, F., Li, D., Vacca, J., Kaushansky, N., Shlush, L., Oren, M., Levine, R., Pikarsky, E., Snir-Alkalay, I., Ben-Neriah, Y.
Cell
HeaderTransferase
Released2018-07-04
Resolution3.170
CATH Insert Date02 Sep, 2018

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2018 Chopped
B 02 Sep, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6gzhA01 03 Sep, 2018 3.30.200.20 Assigned
6gzhA02 03 Sep, 2018 1.10.510.10 Assigned
6gzhB01 03 Sep, 2018 1.10.472.10 Assigned
6gzhB02 03 Sep, 2018 1.10.472.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60563 CCNT1_HUMAN Homo sapiens Cyclin-T1
P50750 CDK9_HUMAN Homo sapiens Cyclin-dependent kinase 9