PDB Information

PDB6GJ4
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Structure-activity relationships, biological evaluation and structural studies of novel pyrrolonaphthoxazepines as antitumor agents.
Brindisi, M., Ulivieri, C., Alfano, G., Gemma, S., de Asis Balaguer, F., Khan, T., Grillo, A., Chemi, G., Menchon, G., Prota, A.E., Olieric, N., Lucena-Agell, D., Barasoain, I., Diaz, J.F., Nebbioso, A., Conte, M., Lopresti, L., Magnano, S., Amet, R., Kinsella, P., Zisterer, D.M., Ibrahim, O., O'Sullivan, J., Morbidelli, L., Spaccapelo, R., Baldari, C., Butini, S., Novellino, E., Campiani, G., Altucci, L., Steinmetz, M.O., Brogi, S.
Eur J Med Chem
HeaderCell Cycle
Released2018-05-16
Resolution2.400
CATH Insert Date16 Dec, 2018

PDB Images (23)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped
B 16 Dec, 2018 Chopped
C 16 Dec, 2018 Chopped
D 16 Dec, 2018 Chopped
E 16 Dec, 2018 Chopped
F 16 Dec, 2018 Chopped

CATH Domains (16)

Domain ID Date inserted into CATH Superfamily CATH Status
6gj4A01 28 Feb, 2019 3.40.50.1440 Assigned
6gj4A02 28 Feb, 2019 3.30.1330.20 Assigned
6gj4A03 28 Feb, 2019 1.10.287.600 Assigned
6gj4B01 28 Feb, 2019 3.40.50.1440 Assigned
6gj4B02 28 Feb, 2019 3.30.1330.20 Assigned
6gj4B03 28 Feb, 2019 1.10.287.600 Assigned
6gj4C01 28 Feb, 2019 3.40.50.1440 Assigned
6gj4C02 28 Feb, 2019 3.30.1330.20 Assigned
6gj4C03 28 Feb, 2019 1.10.287.600 Assigned
6gj4D01 28 Feb, 2019 3.40.50.1440 Assigned
6gj4D02 28 Feb, 2019 3.30.1330.20 Assigned
6gj4D03 28 Feb, 2019 1.10.287.600 Assigned
6gj4E01 28 Feb, 2019 6.10.280.30 Assigned
6gj4F01 28 Feb, 2019 3.40.50.11480 Assigned
6gj4F02 28 Feb, 2019 3.30.470.20 Assigned
6gj4F03 28 Feb, 2019 Holding pen

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P63043 STMN4_RAT Rattus norvegicus Stathmin-4
E1BQ43 E1BQ43_CHICK Gallus gallus Uncharacterized protein
Q6B856 TBB2B_BOVIN Bos taurus Tubulin beta-2B chain
P81947 TBA1B_BOVIN Bos taurus Tubulin alpha-1B chain
Q6B856 TBB2B_BOVIN Bos taurus Tubulin beta-2B chain
P81947 TBA1B_BOVIN Bos taurus Tubulin alpha-1B chain