PDB Information

PDB6G8M
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae
Gene SourceSaccharomyces cerevisiae (strain ATCC 204508 / S288c)
Primary Citation
Design, synthesis, and evaluation of cystargolide-based beta-lactones as potent proteasome inhibitors.
Niroula, D., Hallada, L.P., Le Chapelain, C., Ganegamage, S.K., Dotson, D., Rogelj, S., Groll, M., Tello-Aburto, R.
Eur J Med Chem
HeaderHydrolase
Released2018-04-09
Resolution2.700
CATH Insert Date16 Sep, 2018

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 16 Sep, 2018 Chopped
A 16 Sep, 2018 Chopped
b 16 Sep, 2018 Chopped
B 16 Sep, 2018 Chopped
C 16 Sep, 2018 Chopped
D 16 Sep, 2018 Chopped
E 16 Sep, 2018 Chopped
F 16 Sep, 2018 Chopped
G 16 Sep, 2018 Chopped
H 16 Sep, 2018 Chopped
I 16 Sep, 2018 Chopped
J 16 Sep, 2018 Chopped
K 16 Sep, 2018 Chopped
L 16 Sep, 2018 Chopped
M 16 Sep, 2018 Chopped
N 16 Sep, 2018 Chopped
O 16 Sep, 2018 Chopped
P 16 Sep, 2018 Chopped
Q 16 Sep, 2018 Chopped
R 16 Sep, 2018 Chopped
S 16 Sep, 2018 Chopped
T 16 Sep, 2018 Chopped
U 16 Sep, 2018 Chopped
V 16 Sep, 2018 Chopped
W 16 Sep, 2018 Chopped
X 16 Sep, 2018 Chopped
Y 16 Sep, 2018 Chopped
Z 16 Sep, 2018 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
6g8ma00 17 Sep, 2018 3.60.20.10 Assigned
6g8mA00 17 Sep, 2018 3.60.20.10 Assigned
6g8mb00 17 Sep, 2018 3.60.20.10 Assigned
6g8mB00 17 Sep, 2018 3.60.20.10 Assigned
6g8mC00 17 Sep, 2018 3.60.20.10 Assigned
6g8mD00 17 Sep, 2018 3.60.20.10 Assigned
6g8mE00 17 Sep, 2018 3.60.20.10 Assigned
6g8mF00 17 Sep, 2018 3.60.20.10 Assigned
6g8mG00 17 Sep, 2018 3.60.20.10 Assigned
6g8mH00 17 Sep, 2018 3.60.20.10 Assigned
6g8mI00 17 Sep, 2018 3.60.20.10 Assigned
6g8mJ00 17 Sep, 2018 3.60.20.10 Assigned
6g8mK00 17 Sep, 2018 3.60.20.10 Assigned
6g8mL00 17 Sep, 2018 3.60.20.10 Assigned
6g8mM00 17 Sep, 2018 3.60.20.10 Assigned
6g8mN00 17 Sep, 2018 3.60.20.10 Assigned
6g8mO00 17 Sep, 2018 3.60.20.10 Assigned
6g8mP00 17 Sep, 2018 3.60.20.10 Assigned
6g8mQ00 17 Sep, 2018 3.60.20.10 Assigned
6g8mR00 17 Sep, 2018 3.60.20.10 Assigned
6g8mS00 17 Sep, 2018 3.60.20.10 Assigned
6g8mT00 17 Sep, 2018 3.60.20.10 Assigned
6g8mU00 17 Sep, 2018 3.60.20.10 Assigned
6g8mV00 17 Sep, 2018 3.60.20.10 Assigned
6g8mW00 17 Sep, 2018 3.60.20.10 Assigned
6g8mX00 17 Sep, 2018 3.60.20.10 Assigned
6g8mY00 17 Sep, 2018 3.60.20.10 Assigned
6g8mZ00 17 Sep, 2018 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7