PDB Information

PDB6G0W
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design, synthesis and evaluation of potent and selective inhibitors of mono-(ADP-ribosyl)transferases PARP10 and PARP14.
Holechek, J., Lease, R., Thorsell, A.G., Karlberg, T., McCadden, C., Grant, R., Keen, A., Callahan, E., Schuler, H., Ferraris, D.
Bioorg. Med. Chem. Lett.
HeaderTransferase
Released2018-03-20
Resolution2.340
CATH Insert Date03 Jun, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6g0wA00 29 Jun, 2018 3.90.228.10 Assigned
6g0wB00 29 Jun, 2018 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q460N5 PAR14_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP14
Q460N5 PAR14_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP14