PDB Information

PDB6FTN
MethodX-RAY DIFFRACTION
Host OrganismInsect cell expression vector pTIE1
Gene SourceMus musculus
Primary Citation
Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3-Kinase (PI3K)-gamma Inhibitors.
Pemberton, N., Mogemark, M., Arlbrandt, S., Bold, P., Cox, R.J., Gardelli, C., Holden, N.S., Karabelas, K., Karlsson, J., Lever, S., Li, X., Lindmark, H., Norberg, M., Perry, M.W.D., Petersen, J., Rodrigo Blomqvist, S., Thomas, M., Tyrchan, C., Westin Eriksson, A., Zlatoidsky, P., Oster, L.
J. Med. Chem.
HeaderTransferase
Released2018-02-22
Resolution2.000
CATH Insert Date06 Jul, 2018

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 06 Jul, 2018 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform