PDB Information

PDB6EZG
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Novel multitarget-directed ligands targeting acetylcholinesterase and sigma1receptors as lead compounds for treatment of Alzheimer's disease: Synthesis, evaluation, and structural characterization of their complexes with acetylcholinesterase.
Lalut, J., Santoni, G., Karila, D., Lecoutey, C., Davis, A., Nachon, F., Silman, I., Sussman, J., Weik, M., Maurice, T., Dallemagne, P., Rochais, C.
Eur J Med Chem
HeaderHydrolase
Released2017-11-15
Resolution2.200
CATH Insert Date16 Dec, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped
B 16 Dec, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6ezgA00 28 Feb, 2019 3.40.50.1820 Assigned
6ezgB00 28 Feb, 2019 3.40.50.1820 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04058 ACES_TETCF Tetronarce californica Acetylcholinesterase
P04058 ACES_TETCF Tetronarce californica Acetylcholinesterase