PDB Information

PDB6ELA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies.
Nuti, E., Cuffaro, D., Bernardini, E., Camodeca, C., Panelli, L., Chaves, S., Ciccone, L., Tepshi, L., Vera, L., Orlandini, E., Nencetti, S., Stura, E.A., Santos, M.A., Dive, V., Rossello, A.
J. Med. Chem.
HeaderHydrolase
Released2017-09-28
Resolution1.490
CATH Insert Date03 Jun, 2018

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped
C 03 Jun, 2018 Chopped
D 03 Jun, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6elaA00 29 Jun, 2018 3.40.390.10 Assigned
6elaB00 29 Jun, 2018 3.40.390.10 Assigned
6elaC00 29 Jun, 2018 3.40.390.10 Assigned
6elaD00 29 Jun, 2018 3.40.390.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase