PDB Information

PDB6EK3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10.
Murthy, S., Desantis, J., Verheugd, P., Maksimainen, M.M., Venkannagari, H., Massari, S., Ashok, Y., Obaji, E., Nkizinkinko, Y., Luscher, B., Tabarrini, O., Lehtio, L.
Eur J Med Chem
HeaderTransferase
Released2017-09-25
Resolution1.600
CATH Insert Date29 Jul, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jul, 2018 Chopped
B 29 Jul, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6ek3A00 30 Jul, 2018 3.90.228.10 Assigned
6ek3B00 30 Jul, 2018 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q460N3 PAR15_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP15
Q460N3 PAR15_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP15