PDB Information

PDB6EIQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Novel Scaffolds for Dual Specificity Tyrosine-Phosphorylation-Regulated Kinase (DYRK1A) Inhibitors.
Czarna, A., Wang, J., Zelencova, D., Liu, Y., Deng, X., Choi, H.G., Zhang, T., Zhou, W., Chang, J.W., Kildalsen, H., Seternes, O.M., Gray, N.S., Engh, R.A., Rothweiler, U.
J. Med. Chem.
HeaderTransferase
Released2017-09-19
Resolution2.300
CATH Insert Date02 Sep, 2018

PDB Images (5)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2018 Holding pen
B 02 Sep, 2018 Holding pen
C 02 Sep, 2018 Holding pen
D 02 Sep, 2018 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A