PDB 6cq5
PDB Information
| PDB | 6CQ5 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Design, synthesis, and biological activity of substituted 2-amino-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid derivatives as inhibitors of the inflammatory kinases TBK1 and IKK epsilon for the treatment of obesity.
Bioorg. Med. Chem.
|
| Header | Transferase |
| Released | 2018-03-14 |
| Resolution | 3.350 |
| CATH Insert Date | 16 Dec, 2018 |
PDB Images (6)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Dec, 2018 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6cq5A01 | 28 Feb, 2019 | 3.30.200.20 | Assigned |
| 6cq5A02 | 28 Feb, 2019 | 1.10.510.10 | Assigned |
| 6cq5A03 | 28 Feb, 2019 | 3.10.20.90 | Assigned |
| 6cq5A04 | 28 Feb, 2019 | 1.20.1270.420 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9UHD2 | TBK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase TBK1 |
