PDB Information

PDB6BYZ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Substrate-selective inhibitors that reprogram the activity of insulin-degrading enzyme.
Maianti, J.P., Tan, G.A., Vetere, A., Welsh, A.J., Wagner, B.K., Seeliger, M.A., Liu, D.R.
Nat.Chem.Biol.
HeaderHydrolase/Inhibitor
Released2017-12-21
Resolution2.960
CATH Insert Date07 Apr, 2019

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 07 Apr, 2019 Chopped
B 07 Apr, 2019 Chopped
D 07 Apr, 2019 Rejected
E 07 Apr, 2019 Rejected

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
6byzA01 08 Apr, 2019 3.30.830.10 Assigned
6byzA02 08 Apr, 2019 3.30.830.10 Assigned
6byzA03 08 Apr, 2019 3.30.830.10 Assigned
6byzA04 08 Apr, 2019 3.30.830.10 Assigned
6byzB01 08 Apr, 2019 3.30.830.10 Assigned
6byzB02 08 Apr, 2019 3.30.830.10 Assigned
6byzB03 08 Apr, 2019 3.30.830.10 Assigned
6byzB04 08 Apr, 2019 3.30.830.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme