PDB 6b4l
PDB Information
PDB | 6B4L |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Structure-guided design of a series of MCL-1 inhibitors with high affinity and selectivity.
J. Med. Chem.
|
Header | Signaling Protein/Inhibitor |
Released | 2017-09-26 |
Resolution | 2.250 |
CATH Insert Date | 14 Nov, 2017 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 14 Nov, 2017 | Chopped |
B | 14 Nov, 2017 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
6b4lA01 | 10 Dec, 2017 | 1.10.437.10 | Assigned |
6b4lB01 | 10 Dec, 2017 | 1.10.437.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q07820 | MCL1_HUMAN | Homo sapiens | Induced myeloid leukemia cell differentiation protein Mcl-1 |
Q07820 | MCL1_HUMAN | Homo sapiens | Induced myeloid leukemia cell differentiation protein Mcl-1 |