PDB 6alc

PDB Information

PDB6ALC
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and synthesis of a biaryl series as inhibitors for the bromodomains of CBP/P300.
Lai, K.W., Romero, F.A., Tsui, V., Beresini, M.H., de Leon Boenig, G., Bronner, S.M., Chen, K., Chen, Z., Choo, E.F., Crawford, T.D., Cyr, P., Kaufman, S., Li, Y., Liao, J., Liu, W., Ly, J., Murray, J., Shen, W., Wai, J., Wang, F., Zhu, C., Zhu, X., Magnuson, S.
Bioorg. Med. Chem. Lett.
HeaderProtein Binding/Inhibitor
Released2017-08-07
Resolution1.390
CATH Insert Date12 Aug, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 12 Aug, 2018 Chopped
B 12 Aug, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6alcA00 13 Aug, 2018 1.20.920.10 Assigned
6alcB00 13 Aug, 2018 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein