PDB 6afr
PDB Information
| PDB | 6AFR |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli K-12 |
| Gene Source | Homo sapiens |
| Primary Citation | Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors
Eur J Med Chem
|
| Header | Signaling Protein/Inhibitor |
| Released | 2018-08-08 |
| Resolution | 2.000 |
| CATH Insert Date | 16 Dec, 2018 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Dec, 2018 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6afrA01 | 28 Feb, 2019 | 1.20.920.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
