PDB Information

PDB5ZG0
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
TAK-137, an AMPA-R potentiator with little agonistic effect, has a wide therapeutic window.
Kunugi, A., Tanaka, M., Suzuki, A., Tajima, Y., Suzuki, N., Suzuki, M., Nakamura, S., Kuno, H., Yokota, A., Sogabe, S., Kosugi, Y., Awasaki, Y., Kaku, T., Kimura, H.
Neuropsychopharmacology
HeaderTransport Protein
Released2018-03-07
Resolution1.580
CATH Insert Date20 Jan, 2019

PDB Images (19)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 20 Jan, 2019 Chopped
B 20 Jan, 2019 Chopped
C 20 Jan, 2019 Chopped
D 20 Jan, 2019 Chopped
E 20 Jan, 2019 Chopped
F 20 Jan, 2019 Chopped

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
5zg0A01 21 Jan, 2019 3.40.190.10 Assigned
5zg0A02 21 Jan, 2019 3.40.190.10 Assigned
5zg0B01 21 Jan, 2019 3.40.190.10 Assigned
5zg0B02 21 Jan, 2019 3.40.190.10 Assigned
5zg0C01 21 Jan, 2019 3.40.190.10 Assigned
5zg0C02 21 Jan, 2019 3.40.190.10 Assigned
5zg0D01 21 Jan, 2019 3.40.190.10 Assigned
5zg0D02 21 Jan, 2019 3.40.190.10 Assigned
5zg0E01 21 Jan, 2019 3.40.190.10 Assigned
5zg0E02 21 Jan, 2019 3.40.190.10 Assigned
5zg0F01 21 Jan, 2019 3.40.190.10 Assigned
5zg0F02 21 Jan, 2019 3.40.190.10 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2